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Browse somatic cancers
by tissues or terms ...
NCI-60 cancer cell lines
Browse cancer-related
KEGG pathways ...
....
Find target by gene identifier
Find targets by list of
gene identifiers
Browse cancer-related
KEGG pathways
Find targets by NCI-60
gene expression ...
... using a gene identifier
... using a KEGG pathway
... using significant
gene expression in 1 to 7
single NCI-60 cell lines
Find targets by
differential gene expression ...
... within 2 NCI-60 cell lines
... from one own/external expression data set against one NCI-60 cell line
... from one own/external expression data set to
determine the the closest NCI-60 cancer cell line
... from two own/external expression data sets
(e.g., cancer/normal)
... from own/external expression data
using pre-calculated ratios
Connectivity Map ...
... explore drug influence on
differential gene expression
Find drugs ...
... by identifier
... by chemical property
... by structure
Find drugs by similarity
in growth activity of NCI-60 cancer cell lines (cellular fingerprints) ...
... using a compound identifier
... of a compound group
... manually defining a
cellular fingerprint
... defining and searching by a compound structure
Find drugs most
biologically active against
a NCI-60 cancer cell line
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doi: 10.1093/nar/gkq910
Target search: 1 gene found
Retinoic acid receptor alpha
(ENSG00000131759 - RARA - P10276 A8K840 A8MUP8 B3KUX3 B4E1J4 B8Y636 C9JS86 Q658K5 Q6I9R7)
Cancer relevance of RARA (ENSG00000131759)
Cancer-related Pathways for KEGG gene
5914
Acute myeloid leukemia
Cancer-related Literature
180240
(gene)
612376
(phenotype)
Cancer Types
from drug target interaction databases
bone, brain, leukemia, lung, neck, skin, various
Connectivity Map
Drug Treatment - Expression Data
ENSG00000131759
NCI-60
expression for ENSG00000131759
cancer cell lines
216300_x_at
203750_s_at
203749_s_at
211605_s_at
mean
NCI-60
expression of PPI partners of ...
ENSG00000131759
Drugs interacting with RARA (ENSG00000131759)
Acitretin
DrugBank
PMID
(9 citations)
adapalene
DrugBank
PMID
(9 citations)
alitretinoin
CTD
PMID
(5 citations)
TTD
drug ID
DAP000275
DrugBank
PMID
(9 citations)
Am 80
TTD
drug ID
DAP000461
DrugBank
PMID
(9 citations)
arsenic trioxide
CTD
PMID
(3 citations)
caffeic acid phenethyl ester
CTD
PMID
16766008
docetaxel
CancerResource
PMID
16129372
Etretinate
DrugBank
PMID
(9 citations)
Oleic Acid
PDB
structure
1DKF
tazarotene
DrugBank
PMID
(9 citations)
wortmannin
CancerResource
PMID
12834623
LG100268
TTD
drug ID
DCL000277
Drug interactions of PPI partners of ...
P10276
← explore drug target interactions of protein-protein-interaction partners
Protein information from multiple resources on RARA (ENSG00000131759)
Target protein
P10276 - RARA_HUMAN
Description
Retinoic acid receptor alpha
Synonyms
Nuclear receptor subfamily 1 group B member 1 - RAR-alpha
virtual access to literature search results
P10276
Protein complex association
CBP-RARA-RXRA-DNA complex, ligand stimulated
Protein Identifier
RARA_HUMAN
Protein Accession Number
P10276
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein IDs
ENSP00000254066
,
ENSP00000377649
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000394089
Structure Information
1DSZ
-
1DKF
Domain families
Hormone_recep
-
zf-C4
Gene ID
5914
virtual access to biological pathways
P10276
Protein-protein interaction (PPI) partners of ...
P10276
← Q13472 P29590 P10276 Q05516 P50120
Target protein
A8K840 - A8K840_HUMAN
virtual access to literature search results
A8K840
Protein Identifier
A8K840_HUMAN
Protein Accession Number
A8K840
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein IDs
ENSP00000254066
,
ENSP00000377649
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000394089
,
ENST00000394089
Domain families
Hormone_recep
-
zf-C4
virtual access to biological pathways
A8K840
Target protein
A8MUP8 - A8MUP8_HUMAN
virtual access to literature search results
A8MUP8
Protein Identifier
A8MUP8_HUMAN
Protein Accession Number
A8MUP8
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000377648
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000394086
Domain families
Hormone_recep
-
zf-C4
virtual access to biological pathways
A8MUP8
Target protein
B3KUX3 - B3KUX3_HUMAN
virtual access to literature search results
B3KUX3
Protein Identifier
B3KUX3_HUMAN
Protein Accession Number
B3KUX3
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000377648
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000394086
Domain families
Hormone_recep
-
zf-C4
virtual access to biological pathways
B3KUX3
Target protein
B4E1J4 - B4E1J4_HUMAN
virtual access to literature search results
B4E1J4
Protein Identifier
B4E1J4_HUMAN
Protein Accession Number
B4E1J4
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000399453
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000394086
Domain family
zf-C4
virtual access to biological pathways
B4E1J4
Target protein
B8Y636 - B8Y636_HUMAN
virtual access to literature search results
B8Y636
Protein Identifier
B8Y636_HUMAN
Protein Accession Number
B8Y636
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000389993
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000425707
Domain family
Hormone_recep
virtual access to biological pathways
B8Y636
Target protein
C9JS86 - C9JS86_HUMAN
virtual access to literature search results
C9JS86
Protein Identifier
C9JS86_HUMAN
Protein Accession Number
C9JS86
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000388570
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000425707
Domain family
Hormone_recep
virtual access to biological pathways
C9JS86
Target protein
Q658K5 - Q658K5_HUMAN
virtual access to literature search results
Q658K5
Protein Identifier
Q658K5_HUMAN
Protein Accession Number
Q658K5
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein ID
ENSP00000316769
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000319149
Domain families
Hormone_recep
-
zf-C4
virtual access to biological pathways
Q658K5
Target protein
Q6I9R7 - Q6I9R7_HUMAN
virtual access to literature search results
Q6I9R7
Protein Identifier
Q6I9R7_HUMAN
Protein Accession Number
Q6I9R7
Gene Symbol
RARA
Gene ID
ENSG00000131759
Protein IDs
ENSP00000254066
,
ENSP00000377649
Variations (Gene as map --- transcript as list)
ENSG00000131759
---
ENST00000319149
,
ENST00000394089
Domain families
Hormone_recep
-
zf-C4
Gene ID
5914
virtual access to biological pathways
Q6I9R7